|
---|
Angiopoietin | - Agonis: Angiopoietin 1
- Angiopoietin 4
- Antagonis: Angiopoietin 2
- Angiopoietin 3
- Perencat kinase: Altiratinib
- CE-245677
- Rebastinib
- Antibodi: Evinasumab (melawan angiopoietin 3)
- Nesvasumab (melawan angiopoietin 2)
|
---|
CNTF | - Agonis: Aksokina
- CNTF
- Dapiklermin
|
---|
EGF (ErbB) | EGF (ErbB1/HER1) | - Agonis: Amfiregulin
- Betaselulin
- EGF (urogastron)
- Epigen
- Epiregulin
- Faktor pertumbuhan seperti EGF pengikat heparin (HB-EGF)
- Murodermin
- Nepidermin
- Faktor pertumbuhan transformasi alfa (TGFα)
- Perencat kinase: Afatinib
- Agerafenib
- Brigatinib
- Dakomitinib
- Erlotinib
- Gefitinib
- Grandinin
- Ikotinib
- Kanertinib
- Lapatinib
- Neratinib
- Osimertinib
- Vandetanib
- WHI-P 154
- Antibodi: Depatuksizumab
- Depatuksizumab mafodotin
- Futuksimab
- Imgatuzumab
- Matuzumab
- Nesitumumab
- Nimotuzumab
- Panitumumab
- Setuksimab
- Zalutumumab
|
---|
ErbB2/HER2 | - Agonis: Tidak diketahui/tiada
- Antibodi: Ertumaksomab
- Pertuzumab
- Trastuzumab
- Trastuzumab derukstekan
- Trastuzumab duokarmazina
- Trastuzumab emtansina
- Perencat kinase: Afatinib
- Lapatinib
- Mubritinib
- Neratinib
- Tukatinib
|
---|
ErbB3/HER3 | - Agonis: Neuregulin (heregulin) (1, 2, 6 (neuroglikan C))
- Antibodi: Duligotumab
- Patritumab
- Seribantumab
|
---|
ErbB4/HER4 | - Agonis: Betaselulin
- Epigen
- Faktor pertumbuhan seperti EGF pengikat heparin (HB-EGF)
- Neuregulin (heregulin) (1, 2, 3, 4, 5 (tomoregulin, TMEFF))
|
---|
|
---|
FGF | FGFR1 | - Agonis: Ersofermin
- FGF (1, 2 (bFGF), 3, 4, 5, 6, 8, 10 (KGF2), 20)
- Repifermin
- Selperkatinib
- Trafermin
- Velafermin
|
---|
FGFR2 | - Agonis: Ersofermin
- FGF (1, 2 (bFGF), 3, 4, 5, 6, 7 (KGF), 8, 9, 10 (KGF2), 17, 18, 22)
- Palifermin
- Repifermin
- Selperkatinib
- Sprifermin
- Trafermin
- Antibodi: Aprutumab
- Aprutumab iksadotin
- Perencat kinase: Infigratinib
|
---|
FGFR3 | - Agonis: Ersofermin
- FGF (1, 2 (bFGF), 4, 8, 9, 18, 23)
- Selperkatinib
- Sprifermin
- Trafermin
- Antibodi: Burosumab (melawan FGF23)
|
---|
FGFR4 | - Agonis: Ersofermin
- FGF (1, 2 (bFGF), 4, 6, 8, 9, 19)
- Trafermin
|
---|
Tidak dikelaskan | |
---|
|
---|
HGF (c-Met) | - Agonis: Fosgonimeton
- Faktor pertumbuhan hepatosit
- Penguat: Diheksa (PNB-0408)
- Perencat kinase: Altiratinib
- AM7
- AMG-458
- Amuvatinib
- BMS-777607
- Foretinib
- Golvatinib
- INCB28060
- JNJ-38877605
- K252a
- Kabozantinib
- Kapmatinib
- Krizotinib
- MK-2461
- PF-04217903
- PF-2341066
- PHA-665752
- SU-11274
- Tivantinib
- Volitinib
- Antibodi: Emibetuzumab
- Fiklatuzumab
- Flanvotumab
- Onartuzumab
- Rilotumumab
- Telisotuzumab
- Telisotuzumab vedotin
|
---|
IGF | IGF-1 | - Perencat kinase: BMS-754807
- Linsitinib
- NVP-ADW742
- NVP-AEW541
- OSl-906
- Antibodi: AVE-1642
- Dalotuzumab
- Figitumumab
- Ganitumab
- Robatumumab
- R1507
- Siksutumumab
- Teprotumumab
- Xentuzumab (melawan IGF-1 dan IGF-2)
|
---|
IGF-2 | - Antibodi: Dusigitumab
- Xentuzumab (melawan IGF-1 and IGF-2)
|
---|
Lain-lain | - Protein pengikat: IGFBP (1, 2, 3, 4, 5, 6, 7)
- Produk pengurai/terbitan dengan sasaran tidak diketahui: Glipromat (GPE, (1-3)IGF-1)
- Trofinetida
|
---|
|
---|
LNGF (p75NTR) | - Agonis: BDNF
- BNN-20
- BNN-27
- DHEA
- DHEA-S
- NGF
- NT-3
- NT-4
- Senegermin
- Antibodi: Melawan NGF: ABT-110 (PG110)
- ASP-6294
- Fasinumab
- Frunevetmab
- Fulranumab
- MEDI-578
- Ranevetmab
- Tanezumab
- Aptamer: Melawan NGF: RBM-004
- Reseptor samaran: LEVI-04 (p75NTR-Fc)
|
---|
PDGF | - Perencat kinase: Agerafenib
- Avapritinib
- Aksitinib
- Krenolanib
- Kuizartinib
- Imatinib
- Lenvatinib
- Masitinib
- Motesanib
- Nintedanib
- Pazopanib
- Radotinib
- Ripretinib
- Sunitinib
- Sorafenib
- Toseranib
- Antibodi: Olaratumab
- Ramusirumab
- Tovetumab
|
---|
RET (GFL) | GFRα1 | - Agonis: Faktor neutrotofik terbitan barisan sel glia (GDNF)
- Liatermin
- Perencat kinase: Vandetanib
|
---|
GFRα2 | - Perencat kinase: Vandetanib
|
---|
GFRα3 | - Perencat kinase: Vandetanib
|
---|
GFRα4 | - Perencat kinase: Vandetanib
|
---|
Tidak dikelaskan | - Perencat kinase: Agerafenib
|
---|
|
---|
SCF (c-Kit) | - Agonis: Ansestim
- Faktor sel tunjang
- Perencat kinase: Agerafenib
- Axitinib
- Dasatinib
- Imatinib
- Masitinib
- Nilotinib
- Pazopanib
- Quizartinib
- Sorafenib
- Sunitinib
- Toceranib
|
---|
TGFβ | |
---|
Trk | TrkA | - Agonis: Amitriptilina
- BNN-20
- BNN-27
- DHEA
- DHEA-S
- Gambogik amida
- NGF
- Senegermin
- Tavilermida
- Pemodulat alosterik negatif: VM-902A
- Perencat kinase: Altiratinib
- AZD-6918
- CE-245677
- CH-7057288
- DS-6051
- Entrektinib
- GZ-389988
- K252a
- Larotrektinib
- Lestaurtinib
- Milsiklib
- ONO-4474
- ONO-5390556
- PLX-7486
- Rebastinib
- SNA-120 (K252a berpegil))
- Antibodi: Melawan TrkA: GBR-900; Melawan NGF: ABT-110 (PG110)
- ASP-6294
- Fasinumab
- Frunevetmab
- Fulranumab
- MEDI-578
- Ranevetmab
- Tanezumab
- Aptamer: Melawan NGF: RBM-004
- Reseptor samaran: ReN-1820 (TrkAd5)
|
---|
TrkB | - Agonis: 3,7-DHF
- 3,7,8,2'-THF
- 4'-DMA-7,8-DHF
- 7,3'-DHF
- 7,8-DHF
- 7,8,2'-THF
- 7,8,3'-THF
- Amitriptilina
- BDNF
- BNN-20
- Deoksigedunin
- Deprenil
- Diosmetin
- DMAQ-B1
- HIOC
- LM22A-4
- N-Asetilserotonin
- NT-3
- NT-4
- Norwogonin (5,7,8-THF)
- R7
- R13
- TDP6
- Antagonis: ANA-12
- Siklotraksin B
- Gosipetin (3,5,7,8,3',4'-HHF)
- Perencat kinase: Altiratinib
- AZD-6918
- CE-245677
- CH-7057288
- DS-6051
- Entrektinib
- GZ-389988
- K252a
- Larotrektinib
- Lestaurtinib
- ONO-4474
- ONO-5390556
- PLX-7486
|
---|
TrkC | - Perencat kinase: Altiratinib
- AZD-6918
- CE-245677
- CH-7057288
- DS-6051
- Entrektinib
- GZ-389988
- K252a
- Larotrektinib
- Lestaurtinib
- ONO-4474
- ONO-5390556
- PLX-7486
|
---|
|
---|
VEGF | - Agonis: Faktor pertumbuhan plasenta (PGF)
- Ripretinib
- Telbermin
- VEGF (A, B, C, D (FIGF))
- Pemodulat alosterik: Cyclotraxin B
- Perencat kinase: Agerafenib
- Altiratinib
- Aksitinib
- Frukuintinib
- Kabozantinib
- Lapatinib
- Lenvatinib
- Motesanib
- Nintedanib
- Pazopanib
- Pegaptanib
- Rebastinib
- Regorafenib
- Sediranib
- Semaksanib
- Sorafenib
- Sunitinib
- Toseranib
- Tivozanib
- Vandetanib
- WHI-P 154
- Antibodi: Alasizumab pegol
- Bevasizumab
- Ikrukumab
- Ramukirumab
- Ranibizumab
- Reseptor samaran: Aflibersept
|
---|
Lain-lain | - Faktor pertumbuhan tambahan: Adrenomedulin
- Faktor perangsang koloni (lihat di sini)
- Faktor pertumbuhan tisu penghubung (CTGF)
- Efrin (A1, A2, A3, A4, A5, B1, B2, B3)
- Eritropoietin (lihat di sini)
- Glukosa-6-fosfat isomerase (GPI; PGI, PHI, AMF)
- Faktor pematangan glia (GMF)
- Faktor pertumbuhan terbitan hepatoma (HDGF)
- Interleukin/faktor pertumbuhan sel T (lihat di sini)
- Faktor perencatan leukemia (LIF)
- Protein perangsang makrofaj (MSP; HLP, HGFLP)
- Midkin (NEGF2)
- Faktor perangsang migrasi (MSF; PRG4)
- Onlomodulin
- Peptida pengaktif adenilat siklase pituitari (PACAP)
- Pleiotrofin
- Renalase
- Trombopoietin (lihat di sini)
- Protein pengisyaratan Wnt
- Pemodulat reseptor faktor pertumbuhan tambahan: Serebrolisin (campuran neurotrofin)
|
---|